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Kinase Inhibitor drugs
45 drugs in this FDA established pharmacologic class, sorted by active ingredient
Kinase Inhibitor list
- CalquenceRxacalabrutinib · Kinase Inhibitor · AstraZeneca Pharmaceuticals LP
- GilotrifRxafatinib · Kinase Inhibitor · Boehringer Ingelheim Pharmaceuticals, Inc.
- InlytaRxaxitinib · Kinase Inhibitor · 2 makers
- BosutinibRxKinase Inhibitor · 3 makers
- AlunbrigRxbrigatinib · Kinase Inhibitor · Takeda Pharmaceuticals America, Inc.
- ZykadiaRxceritinib · Kinase Inhibitor · Novartis Pharmaceuticals Corporation
- XalkoriRxcrizotinib · Kinase Inhibitor · Pfizer Laboratories Div Pfizer Inc
- BalversaRxerdafitinib · Kinase Inhibitor · Janssen Products LP
- ErlotinibRxKinase Inhibitor · 6 makers
- EverolimusRxBoxed warningKinase Inhibitor · 9 makers
- AfinitorRxeverolimus · Kinase Inhibitor · Novartis Pharmaceuticals Corporation
- TorpenzRxeverolimus · Kinase Inhibitor · Upsher-Smith Laboratories, LLC
- YulithiraRxeverolimus · Kinase Inhibitor · CivicaScript, LLC
- EverolimusRxBoxed warningeverolimus tablets · Kinase Inhibitor · Breckenridge Pharmaceutical, Inc.
- LytgobiRxfutibatinib · Kinase Inhibitor · TAIHO PHARMACEUTICAL CO., LTD.
- GefitinibRxKinase Inhibitor · 3 makers
- IressaRxgefitinib · Kinase Inhibitor · AstraZeneca Pharmaceuticals LP
- ImbruvicaRxibrutinib · Kinase Inhibitor · Pharmacyclics LLC
- ItovebiRxinavolisib · Kinase Inhibitor · Genentech, Inc.
- VitrakviRxlarotrectinib · Kinase Inhibitor · 2 makers
- LazcluzeRxlazertinib · Kinase Inhibitor · Janssen Biotech, Inc.
- LorbrenaRxlorlatinib · Kinase Inhibitor · 2 makers
- NilotinibRxBoxed warningKinase Inhibitor · 6 makers
- CavhanzaRxBoxed warningnilotinib · Kinase Inhibitor · Cycle Pharmaceuticals Ltd
- DanzitenRxBoxed warningnilotinib · Kinase Inhibitor · Azurity Pharmaceuticals, Inc.
- VonjoRxpacritinib · Kinase Inhibitor · Sobi, Inc.
- IbranceRxpalbociclib · Kinase Inhibitor · 2 makers
- PazopanibRxBoxed warningKinase Inhibitor · 3 makers
- PemazyreRxpemigatinib · Kinase Inhibitor · Incyte Corporation
- GavretoRxBoxed warningpralsetinib · Kinase Inhibitor · Rigel Pharmaceuticals, Inc.
- AugtyroRxrepotrectinib · Kinase Inhibitor · E.R. Squibb & Sons, L.L.C.
- WayrilzRxrilzabrutinib · Kinase Inhibitor · Genzyme Corporation
- QinlockRxripretinib · Kinase Inhibitor · Deciphera Pharmaceuticals, LLC
- JakafiRxruxolitinib · Janus Kinase Inhibitor · Incyte Corporation
- RydaptRxKinase Inhibitor · Novartis Pharmaceuticals Corporation
- KoselugoRxselumetinib · Kinase Inhibitor · AstraZeneca Pharmaceuticals LP
- SirolimusRxBoxed warningKinase Inhibitor · 13 makers
- HyftorRxsirolimus · Kinase Inhibitor · Nobelpharma America, LLC
- SorafenibRxKinase Inhibitor · 5 makers
- NexavarRxsorafenib · Kinase Inhibitor · Bayer HealthCare Pharmaceuticals Inc.
- OjemdaRxtovorafenib · Kinase Inhibitor · Day One Biopharmaceuticals, Inc.
- CaprelsaRxBoxed warningvandetanib · Kinase Inhibitor · Genzyme Corporation
- ZelborafRxvemurafenib · Kinase Inhibitor · Genentech, Inc.
- RomvimzaRxvimseltinib · Kinase Inhibitor · Deciphera Pharmaceuticals, LLC
- HernexeosRxzongertinib · Kinase Inhibitor · Boehringer Ingelheim Pharmaceuticals, Inc.
Frequently asked questions
- What is a kinase inhibitor?
- Kinase Inhibitor is an FDA established pharmacologic class (EPC). Drugs in the same class work in a similar way, but they can differ in uses, dosing and side effects.
- How many kinase inhibitor drugs are there?
- Our data lists 45 FDA-labeled products in this class, counting brand and generic versions separately.
Source: U.S. Food and Drug Administration, openFDA drug labels · Last updated 10/26/2026